PPIDT00048
Drug Information
| Name | Drotrecogin alfa |
|---|---|
| Sequence | LIDGKMTRRGDSPWQVVLLDSKKKLACGAVLIHPSWVLTAAHCMDESKKLLVRLGEYDLRRWEKWELDLDIKEVFVHPNYSKSTTDNDIALLHLAQPATLSQTIVPICLPDSGLAERELNQAGQETLVTGWGYHSSREKEAKRNRTFVLNFIKIPVVPHNECSEVMSNMVSENMLCAGILGDRQDACEGDSGGPMVASFHGTWFLVGLVSWGEGCGLLHNYGVYTKVSRYLDWIHGHIRDKEAPQKSWAP |
| DrugBank_ID | DB00055 |
| Type | biotech |
| Indication | For reduction of mortality in patients with severe sepsis. |
Dosage Forms
| Form | Route | Strength |
|---|---|---|
| Injection, powder, for solution | Intravenous |
20 mg
|
| Injection, powder, for solution | Intravenous |
5 mg
|
| Injection, powder, lyophilized, for solution | Intravenous |
20 mg/10mL
|
| Injection, powder, lyophilized, for solution | Intravenous |
5 mg/2.5mL
|
| Powder, for solution | Intravenous |
|
| Solution | Parenteral |
5 mg
|
| Powder, for solution | Intravenous |
20 mg / vial
|
| Powder, for solution | Intravenous |
5 mg / vial
|
Target Information
| Role | Uniprot_ID | Gene_Name | Entity_Name | Organism | Actions | Internal link |
|---|---|---|---|---|---|---|
| target | P00451 | F8 | Coagulation factor VIII | Homo sapiens | inhibitor | Link |
| target | P12259 | F5 | Coagulation factor V | Homo sapiens | inhibitor | Link |
| target | P05121 | SERPINE1 | Plasminogen activator inhibitor 1 | Homo sapiens | unknown | Link |
| target | P07204 | THBD | Thrombomodulin | Homo sapiens | unknown | Link |
| target | P07225 | PROS1 | Vitamin K-dependent protein S | Homo sapiens | unknown | Link |
| target | P00734 | F2 | Prothrombin | Homo sapiens | unknown | Link |
| target | P02776 | PF4 | Platelet factor 4 | Homo sapiens | unknown | Link |
| target | P05154 | SERPINA5 | Plasma serine protease inhibitor | Homo sapiens | unknown | Link |
| target | P35237 | SERPINB6 | Serpin B6 | Homo sapiens | unknown | Link |
| target | Q9UNN8 | PROCR | Endothelial protein C receptor | Homo sapiens | unknown | Link |