PPIDT00062

Drug Information
NameRituximab
SequenceQVQLQQPGAELVKPGASVKMSCKASGYTFTSYNMHWVKQTPGRGLEWIGAIYPGNGDTSYNQKFKGKATLTADKSSSTAYMQLSSLTSEDSAVYYCARSTYYGGDWYFNVWGAGTTVTVSAASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKAEPKSCDKTHTCPPCPAPELLGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALPAPIEKTISKAKGQPREPQVYTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNHYTQKSLSLSPGK
DrugBank_IDDB00073
Typebiotech
IndicationRituximab is indicated for the treatment of adult patients with relapsed or refractory, low-grade or follicular, CD20-positive, B-cell non-Hodgkin’s Lymphoma (NHL) as a single agent. Also, it is indicated for the treatment of adult patients with previously untreated follicular, CD20-positive, B-cell NHL in combination with first line chemotherapy and, in patients achieving a complete or partial response to a rituximab product in combination with chemotherapy, as single-agent maintenance therapy.[L26641,L42025,L42030,L42035,L42040] Additionally, rituximab is indicated for the treatment of adult patients with non-progressing (including stable disease), low-grade, CD20-positive, B-cell NHL as a single agent after first-line cyclophosphamide, vincristine, and prednisone (CVP) chemotherapy; and previously untreated diffuse large B-cell, CD20-positive NHL in combination with cyclophosphamide, doxorubicin, vincristine, prednisone (CHOP) or other anthracycline-based chemotherapy regimens.[L26641,L42025,L42030,L42035,L42040] Rituximab, in combination with fludarabine and cyclophosphamide (FC), is indicated for the treatment of adult patients with previously untreated and previously treated CD20-positive chronic lymphocytic leukemia (CLL).[L26641,L42025,L42030,L42035,L42040] In combination with methotrexate, rituximab is indicated for the treatment of adult patients with moderately-to severely-active rheumatoid arthritis who have had an inadequate response to one or more TNF antagonist therapies.[L26641,L42025,L42030,L42035] Additionally, rituximab, in combination with glucocorticoids, is indicated for the treatment of adult and pediatric patients 2 years of age and older with Granulomatosis with Polyangiitis (GPA) (Wegener’s Granulomatosis) and Microscopic Polyangiitis (MPA).[L26641,L42025,L42030,L42035] RITUXAN (rituximab injection for intravenous use) is indicated for the treatment of pediatric patients aged 6 months and older with previously untreated, advanced stage, CD20-positive diffuse large B-cell lymphoma (DLBCL), Burkitt lymphoma (BL), Burkitt-like lymphoma (BLL) or mature B-cell acute leukemia (B-AL) in combination with chemotherapy; as well as the treatment of adult patients with moderate to severe pemphigus vulgaris.[L26641] These indications for RITUXAN are not included in the labels of rituximab biosimilar products (rituximab-arrx, rituximab-abbs, rituximab-pvvr).[L42025,L42030,L42035] The combination product RITUXAN HYCELA (rituximab and hyaluronidase human injection, for subcutaneous use) is not indicated for the treatment of non-malignant conditions.[L42040]

Dosage Forms
Form Route Strength
Solution Intravenous
100.0 mg
Solution Intravenous; Subcutaneous
1000000 mg
Solution Parenteral
100 mg
Solution, concentrate Intravenous
50000000 mg
Solution Intravenous
10000000 mg
Injection Intravenous
1400 MG/11.7ML
Injection, solution Subcutaneous
1600 mg
Injection, solution, concentrate Intravenous
10 mg/1ml
Injection, solution, concentrate Intravenous
100 mg
Injection, solution, concentrate Intravenous
500 mg
Solution
10 mg/1ml
Solution Intravenous
100.000 mg
Solution Intravenous
500 mg
Solution Intravenous
50000000 mg
Injection Intravenous
100 mg/10ml
Injection, solution, concentrate Intravenous
100 MG/10ML
Injection, solution Intravenous
120 mg/mL
Injection Intravenous
500 mg/50ml
Injection, solution, concentrate Intravenous
500 MG/50ML
Solution Intravenous
10 mg/ml
Injection Intravenous
10 mg/ml
Solution Intravenous
10 mg
Solution Intravenous
1000000 mg
Injection, solution Subcutaneous
1400 mg
Solution, concentrate Intravenous
10 mg/ml
Solution Subcutaneous
120 mg
Solution Subcutaneous
12000000 mg
Injection; injection, solution, concentrate Intravenous
10 MG/ML
Solution Intravenous
500.000 mg
Injection, solution Intravenous
10 mg/1mL
Solution Intravenous
10 mg / mL
Injection, solution Subcutaneous
Solution Subcutaneous
1400 mg / 11.7 mL
Solution Subcutaneous
1600 mg / 13.4 mL
Injection, solution, concentrate
100 mg/10ml
Injection, solution, concentrate
500 mg/50ml
Solution Intravenous
100 mg/10ml
Solution Intravenous
500 mg/50ml
Solution, concentrate Intravenous
1000000 mg
Injection, solution Intravenous
100 mg/10mL
Injection, solution Intravenous
500 mg/50mL
Injection, solution, concentrate Intravenous; Parenteral
100 MG
Solution, concentrate Intravenous
10 mg
Injection, solution, concentrate Intravenous; Parenteral
500 MG
Solution Intravenous
100 mg / 10 mL
Solution Intravenous
500 mg / 50 mL
10 mg/1ml
Injection, solution
1400 mg/11.7ml
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P11836 MS4A1 B-lymphocyte antigen CD20 Homo sapiens antibody|regulator Link