PPIDT00158

Drug Information
NameRamucirumab
SequenceEVQLVQSGGGLVKPGGSLRLSCAASGFTFSSYSMNWVRQAPGKGLEWVSSISSSSSYIYYADSVKGRFTISRDNAKNSLYLQMNSLRAEDTAVYYCARVTDAFDIWGQGTMVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPELLGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALPAPIEKTISKAKGQPREPQVYTLPPSREEMTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNHYTQKSLSLSPGK
DrugBank_IDDB05578
Typebiotech
IndicationRamucirumab is indicated for the treatment of advanced or metastatic gastric or gastro-esophageal junction adenocarcinoma as a single agent or in combination with [paclitaxel] for patients who progress after prior fluoropyrimidine- or platinum-containing chemotherapy. It is indicated, in combination with [erlotinib], for the first-line treatment of metastatic non-small cell lung cancer with epidermal growth factor exon 19 deletions or exon 21 (L858R) point mutations. It is also indicated in combination with [docetaxel] for the treatment of metastatic non-small cell lung cancer in patients who have progressed following prior platinum-based chemotherapy. Patients who have EGFR or ALK genomic aberrations should also have disease progression following FDA-approved therapy for these aberrations. Ramucirumab, in combination with FOLFIRI ([folinic acid], [fluorouracil], and [irinotecan]), is indicated for the treatment of metastatic colorectal cancer in patients who have progressed following therapy with [bevacizumab], [oxaliplatin], and a fluoropyrimidine. Lastly, ramucirumab is indicated for the treatment of hepatocellular carcinoma in patients with an alpha-fetoprotein level ≥400 ng/mL and have previously been treated with [sorafenib].[L40938]

Dosage Forms
Form Route Strength
Injection Intravenous
10 mg/mL
Injection, solution, concentrate Intravenous; Parenteral
10 MG/ML
Solution Intravenous
10 mg / mL
Solution Intravenous
10 mg/1mL
Solution Intravenous
10.000 mg
Injection Parenteral
100 mg/10ml
Injection, solution, concentrate Intravenous
100 mg/10ml
Injection Parenteral
500 mg/50ml
Injection, solution, concentrate Intravenous
500 mg/50ml
Injection, solution, concentrate Intravenous
10 mg/ml
Solution, concentrate Intravenous
1000000 mg
Injection, solution, concentrate Intravenous
10 mg/1ml
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P35968 KDR Vascular endothelial growth factor receptor 2 Homo sapiens antagonist Link