PPIDT00194

Drug Information
NameTocilizumab
SequenceDIQMTQSPSSLSASVGDRVTITCRASQDISSYLNWYQQKPGKAPKLLIYYTSRLHSGVPSRFSGSGSGTDFTFTISSLQPEDIATYYCQQGNTLPYTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC
DrugBank_IDDB06273
Typebiotech
IndicationTocilizumab is indicated to treat moderate to severe rheumatoid arthritis, giant cell arteritis, systemic sclerosis-associated interstitial lung disease, polyarticular juvenile idiopathic arthritis, systemic juvenile idiopathic arthritis, and cytokine release syndrome.[L12789, L43697, L48385] Tocilizumab is also used to treat coronavirus disease 2019 (COVID-19) in adults who are receiving systemic corticosteroids and require supplemental oxygen, mechanical ventilation, or extracorporeal membrane oxygenation (ECMO).[L40169,L43697,L44483]

Dosage Forms
Form Route Strength
Injection Intravenous
162 mg/0.9ml
Injection Intravenous
20 MG/ML
Injection, solution, concentrate Intravenous
20 mg/1mL
Injection, solution, concentrate Intravenous
400 mg/20mL
Injection, solution, concentrate Intravenous
80 mg/4mL
Solution Intravenous
200 mg / 10 mL
Solution Intravenous
400 mg / 20 mL
Solution Intravenous
80 mg / 4 mL
Solution Subcutaneous
162 mg / 0.9 mL
Injection, solution
162 mg/0.9mL
Injection, solution Subcutaneous
162 mg/0.9mL
Injection, solution Intravenous
Solution Intravenous
20 mg/ml
Solution Intravenous
80 mg
Solution Intravenous
200 mg
Solution Intravenous
20000000 mg
Solution Intravenous
40000000 mg
Solution Intravenous
8000000 mg
Solution Subcutaneous
162 mg
Solution Subcutaneous
16200000 mg
Injection, solution Parenteral; Subcutaneous
162 MG
Injection, solution, concentrate Intravenous
20 MG/ML
Solution Intravenous
80.000 mg
Solution Subcutaneous
162.000 mg
Injection Intravenous
20 mg/1mL
Injection, solution Subcutaneous
162 mg
Injection, solution, concentrate Intravenous
200 mg/10mL
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P08887 IL6R Interleukin-6 receptor subunit alpha Homo sapiens inhibitor|antibody Link
enzyme P08684 CYP3A4 Cytochrome P450 3A4 Homo sapiens inducer Link