PPIDT00228

Drug Information
NamePasireotide
SequenceNot Available
DrugBank_IDDB06663
Typesmall molecule
IndicationFor the treatment of Cushing’s disease, specifically for those patients whom pituitary surgery has not been curative or is not an option.

Dosage Forms
Form Route Strength
Injection Subcutaneous
0.3 mg/1mL
Injection Subcutaneous
0.6 mg/1mL
Injection Subcutaneous
0.9 mg/1mL
Injection, powder, for suspension Intramuscular
10 mg
Injection, powder, for suspension Intramuscular
30 mg
Injection, powder, for suspension Intramuscular; Parenteral
10 MG
Injection, powder, for suspension Intramuscular; Parenteral
20 MG
Injection, powder, for suspension Intramuscular; Parenteral
30 MG
Injection, powder, for suspension Intramuscular; Parenteral
40 MG
Injection, powder, for suspension Intramuscular; Parenteral
60 MG
Solution Subcutaneous
0.3 mg / mL
Solution Subcutaneous
0.6 mg / mL
Solution Subcutaneous
0.9 mg / mL
Solution
0.3 mg/1ml
Solution
0.6 mg/1ml
Solution
0.9 mg/1ml
Injection, powder, for suspension Intramuscular
6000000 mg
Injection Subcutaneous
Injection, solution Subcutaneous
0.3 mg/1ml
Injection Subcutaneous
0.375 mg/ml
Solution Oral
0.3 mg/1ml
Injection, solution Subcutaneous
0.6 mg/1ml
Solution Oral
0.6 mg/1ml
Injection, solution Subcutaneous
0.9 mg/1ml
Solution Oral
0.9 mg/1ml
Injection, powder, for suspension, extended release; kit Intramuscular
10 mg
Injection, powder, for suspension, extended release; kit Intramuscular
20 mg
Injection, powder, for suspension, extended release; kit Intramuscular
30 mg
Injection, powder, for suspension, extended release; kit Intramuscular
40 mg
Injection, powder, for suspension, extended release; kit Intramuscular
60 mg
Injection, powder, for suspension; kit Intramuscular
10 mg/1mL
Injection, powder, for suspension; kit Intramuscular
15 mg/1mL
Injection, powder, for suspension; kit Intramuscular
20 mg/1mL
Injection, powder, for suspension; kit Intramuscular
30 mg/1mL
Injection, powder, for suspension; kit Intramuscular
5 mg/1mL
Kit Intramuscular
5 mg/1mL
Injection, powder, for suspension
10 mg/1vial
Injection, powder, for suspension
20 mg/1vial
Injection, powder, for suspension
30 mg/1vial
Injection, powder, for suspension
40 mg/1vial
Powder, for solution Oral
20 mg
Powder, for solution Oral
40 mg
Powder, for solution Oral
60 mg
Injection, powder, for suspension Intramuscular
20 mg
Injection, powder, for suspension Intramuscular
40 mg
Injection, powder, for suspension Intramuscular
60 mg
Injection, powder, for suspension
60 mg/1vial
Injection, solution Subcutaneous
0.3 mg
Injection, solution Subcutaneous
0.6 mg
Injection, solution Subcutaneous
0.9 mg
Solution Subcutaneous
0.3 mg
Solution Subcutaneous
0.6 mg
Solution Subcutaneous
0.9 mg
Injection, powder, for suspension Intramuscular
2742000 mg
Injection, powder, for suspension Intramuscular
4000000 mg
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P32745 SSTR3 Somatostatin receptor type 3 Homo sapiens inhibitor Link
target P30872 SSTR1 Somatostatin receptor type 1 Homo sapiens inhibitor Link
target P30874 SSTR2 Somatostatin receptor type 2 Homo sapiens inhibitor Link
target P35346 SSTR5 Somatostatin receptor type 5 Homo sapiens inhibitor Link
enzyme P08684 CYP3A4 Cytochrome P450 3A4 Homo sapiens inhibitor Link