PPIDT00241

Drug Information
NameBrentuximab vedotin
SequenceNot Available
DrugBank_IDDB08870
Typebiotech
IndicationBrentuximab vedotin is indicated in adult patients for the treatment of previously untreated stage III or IV classical Hodgkin's lymphoma (cHL) in combination with [doxorubicin], [vinblastine], and [dacarbazine]. It is also indicated for the treatment of cHL post-autologous hematopoietic stem cell transplantation (auto-HSCT) in patients at high risk of relapse or progression. Finally, it may be used in the treatment of adult patients with cHL who have previously failed either auto-HSCT or at least two prior multi-agent chemotherapy regimens if they are not candidates for auto-HSCT.[L39789] Brentuximab vedotin is additionally indicated in the treatment of previously untreated systemic anaplastic large cell lymphoma (sALCL), or other CD30-expressing peripheral T-cell lymphomas (PTCL), in combination with [cyclophosphamide], doxorubicin, and [prednisone]. It may also be used as monotherapy in sALCL after therapeutic failure of a least one prior multi-agent chemotherapy regimen.[L39789] Brentuximab vedotin is also indicated in the treatment of primary cutaneous large anaplastic large cell lymphoma, or CD30-expressing mycosis fungoides, who have received prior systemic therapy.[L39789]

Dosage Forms
Form Route Strength
Injection, powder, for solution Intravenous; Parenteral
50 MG
Injection, powder, lyophilized, for solution Intravenous
50 mg/10.5mL
Powder, for solution Intravenous
50 mg / vial
Injection, solution, concentrate Intravenous
50 mg/1vial
Injection, solution Intravenous
50 mg
Powder Intravenous
50 mg
Injection, powder, for solution Intravenous drip
50 mg
Injection, powder, for solution Intravenous
50 mg
Injection, powder, for solution Intravenous
5000000 mg
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P28908 TNFRSF8 Tumor necrosis factor receptor superfamily member 8 Homo sapiens binder|antibody|regulator Link
enzyme P08684 CYP3A4 Cytochrome P450 3A4 Homo sapiens substrate|inhibitor Link
transporter Q2M3G0 ABCB5 ATP-binding cassette sub-family B member 5 Homo sapiens substrate Link