PPIDT00294

Drug Information
NameRavulizumab
SequenceXVQLVQSGAEVKKPGASVKVSCKASGHIFSNYWIQWVRQAPGQGLEWMGEILPGSGHTEYTENFKDRVTMTRDTSTSTVYMELSSLRSEDTAVYYCARYFFGSSPNWYFDVWGQGTLVTVSSASTKGPSVFPLAPCSRSTSESTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSNFGTQTYTCNVDHKPSNTKVDKTVERKCCVECPPCPAPPVAGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSQEDPEVQFNWYVDGVEVHNAKTKPREEQFNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKGLPSSIEKTISKAKGQPREPQVYTLPPSQEEMTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSRLTVDKSRWQEGNVFSCSVLHEALHSHYTQKSLSLSLG
DrugBank_IDDB11580
Typebiotech
IndicationRavulizumab is indicated for the treatment of adult and pediatric patients one month of age and older with paroxysmal nocturnal hemoglobinuria (PNH).[L39690] It is also indicated for the treatment of adult and pediatric patients one month of age and older with atypical hemolytic uremic syndrome (aHUS) to inhibit complement-mediated thrombotic microangiopathy (TMA). However, the FDA advises against the use of ravulizumab for the treatment of patients with Shiga toxin E. coli related hemolytic uremic syndrome (STEC-HUS).[L39690] Ravulizumab is also indicated for the treatment of adult patients with generalized myasthenia gravis (gMG) who are anti-acetylcholine receptor (AChR) antibody-positive.[L39690,L39700] It is indicated for the treatment of adult patients with neuromyelitis optica spectrum disorder (NMOSD) who are anti-aquaporin-4 (AQP4) antibody positive.[L50396] The European Commission approved ravulizumab for the treatment of paroxysmal nocturnal haemoglobinuria (PNH) in adults and children with a body weight of 10 kg or more with the following conditions: hemolysis with clinical symptoms indicative of high disease activity or clinically stable after having been treated with eculizumab for at least the past six months. Ravulizumab is also indicated for the treatment of hemolytic uremic syndrome (aHUS) in patients with a body weight of 10 kg or more who are either complement inhibitor treatment-naïve or have received [eculizumab] for at least 3 months and have evidence of response to eculizumab.[L39700]

Dosage Forms
Form Route Strength
Injection, solution Subcutaneous
245 mg
Injection, solution, concentrate Intravenous
10 mg / mL
Injection, solution, concentrate Intravenous
1100 mg/11mL
Injection, solution, concentrate Intravenous
1100 MG
Injection, solution, concentrate Intravenous
300 mg/3mL
Injection, solution, concentrate Intravenous
300 mg/30mL
Injection, solution, concentrate Intravenous
300 MG
Kit; solution Subcutaneous
245 mg/3.5mL
Solution Intravenous
1100 mg / 11 mL
Solution Intravenous
300 mg / 3 mL
Solution, concentrate Intravenous
10000000 mg
Injection, solution, concentrate Intravenous
100 mg/mL
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P01031 C5 Complement C5 Homo sapiens inhibitor Link