PPIRE01193

Target Protein Information
Protein_Name Actin-related protein 2/3 complex subunit 4
Protein_Sequence MSNTLRPYLNAVRSTLTASLALEEFSSEIVERQSQPEVEVGRSPEILLKPLVVSRNEQEQCLIESSVNSVRFSIRIKQVDEIERILVRKFMQFLMGRAESFFILRRKPVQGYDISFLITNYHTEEMLKHKLVDFIIEFMEEVDAEISEMKLFLNGRARLVAETYLSCF
Organism_Source Schizosaccharomyces pombe (strain 972 / ATCC 24843)
Functional_Classification actin nucleation complex
Cellular_Localization Cytoplasm
Gene_Names arc4
UniProt_ID Q92352
Protein-Protein Interaction Networks
Peptide Basic Information
Peptide_Name Wsp1p-CA
Peptide_Sequence XXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXX
Peptide_Length 33
Peptide_SMILES NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)NCC(=O)O
Chemical_Modification None
Cyclization_Method None
Linear/Cyclic Linear
N-terminal_Modification Free
C-terminal_Modification Free
Amino_Acid_Distribution
Peptide Physicochemical
Molecular_Weight 1900.73
Aliphatic_Index 0.00000
Aromaticity 0.00000
Average_Rotatable_Bonds 1.96970
Charge_at_pH_7 -0.00202
Isoelectric_Point 6.10000
Number_of_Hydrogen_Bond_Acceptors 34
Number_of_Hydrogen_Bond_Donors 34
Topological_Polar_Surface_Area 994.52000
X_logP_energy -29.25190
Interaction Information
Affinity KD=0.13 uM
Affinity_Assay Isothermal titration calorimetry
PDB_ID None
Type Inhibitor
Structure
Reference Information
Document_Type Research Articles
Title Structural and biochemical characterization of two binding sites for nucleation-promoting factor WASp-VCA on Arp2/3 complex.
Release_Year 2011
PMID 21676862
DOI 10.1073/pnas.1100125108