PPIRE09532

Target Protein Information
Protein_Name Alpha-synuclein
Protein_Sequence MDVFMKGLSKAKEGVVAAAEKTKQGVAEAAGKTKEGVLYVGSKTKEGVVHGVATVAEKTKEQVTNVGGAVVTGVTAVAQKTVEGAGSIAAATGFVKKDQLGKNEEGAPQEGILEDMPVDPDNEAYEMPSEEGYQDYEPEA
Organism_Source Homo sapiens
Functional_Classification presynaptic proteins
Cellular_Localization Cytoplasm
Gene_Names SNCA
UniProt_ID P37840
Protein-Protein Interaction Networks
Peptide Basic Information
Peptide_Name alpha-synuclein fibril fragment(epitope 1-10)
Peptide_Sequence MDVFMKGLSK
Peptide_Length 10
Peptide_SMILES CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@@H](N)CCSC)C(C)C)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)O
Chemical_Modification None
Cyclization_Method None
Linear/Cyclic Linear
N-terminal_Modification Free
C-terminal_Modification Free
Amino_Acid_Distribution
Peptide Physicochemical
Molecular_Weight 1155.44
Aliphatic_Index 68.00000
Aromaticity 0.10000
Average_Rotatable_Bonds 4.10000
Charge_at_pH_7 0.99784
Isoelectric_Point 9.53730
Number_of_Hydrogen_Bond_Acceptors 17
Number_of_Hydrogen_Bond_Donors 15
Topological_Polar_Surface_Area 434.79000
X_logP_energy -2.43110
Interaction Information
Affinity EC50=120 pM
Affinity_Assay ELISA
PDB_ID None
Type Affinity ligand
Structure
Reference Information
Document_Type Research Articles
Title Development of an aggregate-selective, human-derived Alpha-synuclein antibody BIIB054 that ameliorates disease phenotypes in Parkinson's disease models.
Release_Year 2018
PMID 30381260
DOI 10.1016/j.nbd.2018.10.016