PPIRE18889
Target Protein Information
| Protein_Name | None |
|---|---|
| Protein_Sequence | MNKTLIALAVSAAAVATGAYADGINQSGDKAGSTVYSAKGTSLEIGGRAEARLSLKDGKAEDKSRVRLNFLGKAEINDSLYGIGFYEGEFTTADSTATKTDNGSDLDNRYTYAGIGGTYGEVTYGKNDGALGVITDFTDIMSYHGNSAADKIAVADRVDNMLAYKGQFGDLGVKASFRFADRTENTVTDKYEDNGKDGYSLSAIYAFGDTGFNVGAGYADQDEQNEYMLAASYRMENLYFAGLFTDGEKAATNGDYTGYELAAGYKLGQAAFTTTYNNAETNDETSANNFAIDATYYFKPNFRTYISYNFNMIDAGDVLGKVGGNGVATKIDAEDELAIGLRYDF |
| Organism_Source | Vibrio mimicus |
| Functional_Classification | Porins outer membrane diffusion channels |
| Cellular_Localization | Extracellular |
| Gene_Names | ompU |
| UniProt_ID | Q27W35 |
| Protein-Protein Interaction Networks | |
Peptide Basic Information
| Peptide_Name | P2 |
|---|---|
| Peptide_Sequence | SCTSPHCFMWLP |
| Peptide_Length | 12 |
| Peptide_SMILES | CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CS)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CS)NC(=O)[C@@H](N)CO)[C@@H](C)O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N1CCC[C@H]1C(=O)O |
| Chemical_Modification | None |
| Cyclization_Method | None |
| Linear/Cyclic | Linear |
| N-terminal_Modification | Free |
| C-terminal_Modification | Free |
| Amino_Acid_Distribution | |
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Peptide Physicochemical
| Molecular_Weight | 1408.67 |
|---|---|
| Aliphatic_Index | 32.50000 |
| Aromaticity | 0.16667 |
| Average_Rotatable_Bonds | 3.08333 |
| Charge_at_pH_7 | -0.03506 |
| Isoelectric_Point | 7.25316 |
|---|---|
| Number_of_Hydrogen_Bond_Acceptors | 20 |
| Number_of_Hydrogen_Bond_Donors | 18 |
| Topological_Polar_Surface_Area | 471.00000 |
| X_logP_energy | -3.29980 |
Interaction Information
| Affinity | KD=0.81 nM |
|---|---|
| Affinity_Assay | ELISA |
| PDB_ID | None |
| Type | Antagonist |
| Structure | |
Reference Information
| Document_Type | Research Articles |
|---|---|
| Title | Screening a Phage Display Library for Two Novel OmpU-Binding Peptides with Adhesion Antagonistic Activity against Vibrio mimicus |
| Release_Year | 2016 |
| PMID | 27832083 |
| DOI | 10.1371/journal.pone.0165092 |