PPIPT00909
Target Protein Information
| Protein_Name | Ighg protein |
|---|---|
| Protein_Sequence | MDISLSLVFLVLFIKGVQCEVQLVETGGGLVQPGRSLKLSCVASGFTFSSYWMYWIRQAPGKGLEWVSSINTDGGSTYYPDSVKGRFTISRDNAENTVYLQMNSLRSEDTATYYCAKGGEYYGYNYPFDYWGQGVMVTVSSAETTAPSVYPLAPGTALKSNSMVTLGCLVKGYFPEPVTVTWNSGALSSGVHTFPAVLQSGLYTLTSSVTVPSSTWPSQTVTCNVAHPASSTKVDKKIVPRNCGGDCKPCICTGSEVSSVFIFPPKPKDVLTITLTPKVTCVVVDISQDDPEVHFSWFVDDVEVHTAQTRPPEEQFNSTFRSVSELPILHQDWLNGRTFRCKVTSAAFPSPIEKTISKPEGRTQVPHVYTMSPTKEEMTQNEVSITCMVKGFYPPDIYVEWQMNGQPQENYKNTPPTMDTDGSYFLYSKLNVKKEKWQQGNTFTCSVLHEGLHNHHTEKSLSHSPGK |
| Organism_Source | Rattus norvegicus |
| Functional_Classification | Ighg protein |
| Cellular_Localization | Extracellular |
| Gene_Names | Ighg |
| UniProt_ID | Q4VBH1 |
| Protein-Protein Interaction Networks | |
Peptide Basic Information
| Peptide_Name | Peptide hybrid 1a |
|---|---|
| Peptide_Sequence | EDDCAWHLGELVWCT |
| Peptide_Length | 15 |
| Peptide_SMILES | CC(C)C[C@H](NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)[C@H](CS)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@@H](N)CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CS)C(=O)N[C@H](C(=O)O)[C@@H](C)O)C(C)C |
| Chemical_Modification | None |
| Cyclization_Method | Side chain-side chain cyclization; C4<->C14; disulfide bond |
| Linear/Cyclic | Linear |
| N-terminal_Modification | PEGylation |
| C-terminal_Modification | Amide |
| Amino_Acid_Distribution | |
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Peptide Physicochemical
| Molecular_Weight | 1776.96 |
|---|---|
| Aliphatic_Index | 78.00000 |
| Aromaticity | 0.13333 |
| Average_Rotatable_Bonds | 3.53333 |
| Charge_at_pH_7 | -4.03061 |
| Isoelectric_point | 3.73726 |
|---|---|
| Number_of_Hydrogen_Bond_Acceptors | 24 |
| Number_of_Hydrogen_Bond_Donors | 26 |
| Topological_Polar_Surface_Area | 700.41000 |
| X_logP_energy | -4.08180 |
Interaction Information
| Affinity | KD=305 nM |
|---|---|
| Affinity_Assay | Surface Plasmon Resonance |
| PDB_ID | None |
| Type | Affinity ligand |
| Structure | |
Reference Information
| Document_Type | Patent |
|---|---|
| Title | METHOD FOR PREPARING ANTIBODY MONOLAYERS WHICH HAVE CONTROLLED ORIENTATION USING PEPTIDE HYBRID |
| Release_Year | 2010 |
| Patent_ID | US20100209945A1 |