PPIPT00912
Target Protein Information
| Protein_Name | Vimentin |
|---|---|
| Protein_Sequence | MSTRSVSSSSYRRMFGGPGTASRPSSSRSYVTTSTRTYSLGSALRPSTSRSLYASSPGGVYATRSSAVRLRSSVPGVRLLQDSVDFSLADAINTEFKNTRTNEKVELQELNDRFANYIDKVRFLEQQNKILLAELEQLKGQGKSRLGDLYEEEMRELRRQVDQLTNDKARVEVERDNLAEDIMRLREKLQEEMLQREEAENTLQSFRQDVDNASLARLDLERKVESLQEEIAFLKKLHEEEIQELQAQIQEQHVQIDVDVSKPDLTAALRDVRQQYESVAAKNLQEAEEWYKSKFADLSEAANRNNDALRQAKQESTEYRRQVQSLTCEVDALKGTNESLERQMREMEENFAVEAANYQDTIGRLQDEIQNMKEEMARHLREYQDLLNVKMALDIEIATYRKLLEGEESRISLPLPNFSSLNLRETNLDSLPLVDTHSKRTLLIKTVETRDGQVINETSQHHDDLE |
| Organism_Source | Homo sapiens |
| Functional_Classification | Intermediate filament protein |
| Cellular_Localization | Cytoplasm |
| Gene_Names | VIM |
| UniProt_ID | P08670 |
| Protein-Protein Interaction Networks | |
Peptide Basic Information
| Peptide_Name | VMT3 |
|---|---|
| Peptide_Sequence | GGGATRSSAVRXSSVGVLLQDS |
| Peptide_Length | 22 |
| Peptide_SMILES | CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)CNC(=O)CNC(=O)CN)[C@@H](C)O)C(C)C)C(C)C)C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CO)C(=O)O |
| Chemical_Modification | X7=citrulline; X12=citrulline |
| Cyclization_Method | None |
| Linear/Cyclic | Cyclic |
| N-terminal_Modification | biotin |
| C-terminal_Modification | Amide |
| Amino_Acid_Distribution | |
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Peptide Physicochemical
| Molecular_Weight | 2061.24 |
|---|---|
| Aliphatic_Index | 84.09091 |
| Aromaticity | 0.00000 |
| Average_Rotatable_Bonds | 3.13636 |
| Charge_at_pH_7 | 0.99842 |
| Isoelectric_point | 10.39777 |
|---|---|
| Number_of_Hydrogen_Bond_Acceptors | 33 |
| Number_of_Hydrogen_Bond_Donors | 37 |
| Topological_Polar_Surface_Area | 999.99000 |
| X_logP_energy | -17.55486 |
Interaction Information
| Affinity | EC50=72.08 uM |
|---|---|
| Affinity_Assay | ELISA |
| PDB_ID | None |
| Type | Affinity ligand |
| Structure | |
Reference Information
| Document_Type | Patent |
|---|---|
| Title | CITRULLINATED PEPTIDES FOR DIAGNOSING AND PROGNOSING RHEUMATOID ARTHRITIS |
| Release_Year | 2014 |
| Patent_ID | US20140170683A1 |