PPIST03459
Protein Information
| Protein_Chain | A[auth E] |
|---|---|
| Protein_Sequence | VKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKDGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF |
Peptide Information
| Peptide_Chain | B[auth I] |
|---|---|
| Peptide_Sequence | TTYADFIASGRTGRRNAIHD |
| Peptide_Length | 20 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 2UZW |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.20 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Syntheses of Potent, Selective, and Orally Bioavailable Indazole-Pyridine Series of Protein Kinase B/Akt Inhibitors with Reduced Hypotension. |
|---|---|
| Release_Year | 2007 |
| PMID | 17523610 |
| DOI | 10.1021/JM0701019 |