PPIST05114
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | GAMDPRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITITPPDQDDSMECVDSERRPHFPQFDYSASSTA |
Peptide Information
| Peptide_Chain | B[auth C] |
|---|---|
| Peptide_Sequence | GRPRTTSFAE |
| Peptide_Length | 10 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 3MV5 |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.47 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Design of selective, ATP-competitive inhibitors of Akt. |
|---|---|
| Release_Year | 2010 |
| PMID | 20481595 |
| DOI | 10.1021/jm1003842 |