PPIST05116

Protein Information
Protein_Chain A;B;C[auth E]
Protein_Sequence MGSSHHHHHHSSGLVPRGSHMGNAAAAKKGSEQESVKEFLAKAKEDFLKKWESPAQNTAHLDQFERIKTLGTGSFGRVMLVKHKETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF
Peptide Information
Peptide_Chain D[auth I];E[auth J];F[auth K]
Peptide_Sequence TTYADFIASGRTGRRNAIHD
Peptide_Length 20
Non-standard residues No
Interaction Information
PDB_ID 3MVJ
Method X-RAY DIFFRACTION
Resolution 2.49 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title Design of selective, ATP-competitive inhibitors of Akt.
Release_Year 2010
PMID 20481595
DOI 10.1021/jm1003842