PPIST05205
Protein Information
| Protein_Chain | A;C |
|---|---|
| Protein_Sequence | GSHMELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ |
Peptide Information
| Peptide_Chain | B;D |
|---|---|
| Peptide_Sequence | KDHQLLRYLLDKDE |
| Peptide_Length | 14 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 3OKI |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.00 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Discovery of novel and orally active FXR agonists for the potential treatment of dyslipidemia & diabetes |
|---|---|
| Release_Year | 2010 |
| PMID | 21134747 |
| DOI | 10.1016/j.bmcl.2010.11.039 |