PPIST06337

Protein Information
Protein_Chain A;B
Protein_Sequence TALAEMPKRKFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQSTQSK
Peptide Information
Peptide_Chain C;D
Peptide_Sequence PIPAWASGNLLTQAIRQQYYKPIDVDRMYGTIDSPKLEELFNKS
Peptide_Length 44
Non-standard residues No
Interaction Information
PDB_ID 3ZTX
Method X-RAY DIFFRACTION
Resolution 1.95 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title Selective Aurora Kinase Inhibitors Identified Using a Taxol- Induced Checkpoint Sensitivity Screen.
Release_Year 2012
PMID 21992004
DOI 10.1021/CB200305U