PPIST06824
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI |
Peptide Information
| Peptide_Chain | B |
|---|---|
| Peptide_Sequence | VEPQKFAEELIHRLEAVQ |
| Peptide_Length | 18 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 3ZDI |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.65 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | 3,6-Diamino-4-(2-Halophenyl)-2-Benzoylthieno(2,3-B) Pyridine-5-Carbonitriles are Selective Inhibitors of Plasmodium Falciparum Glycogen Synthase Kinase-3 (Pfgsk-3) |
|---|---|
| Release_Year | 2013 |
| PMID | 23214499 |
| DOI | 10.1021/JM301575N |