PPIST07241
Protein Information
| Protein_Chain | A[auth H] |
|---|---|
| Protein_Sequence | IVGGKVCPKGECPWQVLLLVNGAQLCGGTLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTNHDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVLNVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTGIVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP |
Peptide Information
| Peptide_Chain | B[auth L] |
|---|---|
| Peptide_Sequence | ICVNENGGCEQYCSDHTGTKRSCRCHEGYSLLADGVSCTPTVEYPCGKIPILEKR |
| Peptide_Length | 55 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 4ISH |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.82 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Discovery and gram-scale synthesis of BMS-593214, a potent, selective FVIIa inhibitor. |
|---|---|
| Release_Year | 2013 |
| PMID | 23478148 |
| DOI | 10.1016/j.bmcl.2013.02.013 |