PPIST08207

Protein Information
Protein_Chain A;B
Protein_Sequence MHHHHHHGENLYFQGSAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGNS
Peptide Information
Peptide_Chain C[auth D];D[auth E]
Peptide_Sequence SLLKKLLD
Peptide_Length 8
Non-standard residues No
Interaction Information
PDB_ID 4WLB
Method X-RAY DIFFRACTION
Resolution 1.70 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title A reversed sulfonamide series of selective RORc inverse agonists.
Release_Year 2014
PMID 25453817
DOI 10.1016/j.bmcl.2014.10.037