PPIST08573
Protein Information
| Protein_Chain | A;C[auth D] |
|---|---|
| Protein_Sequence | MHHHHHHGENLYFQGSAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTE |
Peptide Information
| Peptide_Chain | B;D[auth E] |
|---|---|
| Peptide_Sequence | AHKILHRLLQE |
| Peptide_Length | 11 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 4WPF |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.20 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Minor Structural Change to Tertiary Sulfonamide RORc Ligands Led to Opposite Mechanisms of Action. |
|---|---|
| Release_Year | 2015 |
| PMID | 25815138 |
| DOI | 10.1021/ml500420y |