PPIST08577
Protein Information
| Protein_Chain | A;B |
|---|---|
| Protein_Sequence | MHHHHHHGENLYFQGSAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGNS |
Peptide Information
| Peptide_Chain | C[auth P] |
|---|---|
| Peptide_Sequence | VERLQIFQHLHPI |
| Peptide_Length | 13 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 4WQP |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.99 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Minor Structural Change to Tertiary Sulfonamide RORc Ligands Led to Opposite Mechanisms of Action. |
|---|---|
| Release_Year | 2015 |
| PMID | 25815138 |
| DOI | 10.1021/ml500420y |