PPIST08908
Protein Information
| Protein_Chain | A;C[auth B] |
|---|---|
| Protein_Sequence | MHHHHHHSSGVDLGTENLYFQSMLNTSGSGTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM |
Peptide Information
| Peptide_Chain | B[auth C];D |
|---|---|
| Peptide_Sequence | KMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPEG |
| Peptide_Length | 49 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 5C5R |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.55 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Fragment-Based Drug Design of Novel Pyranopyridones as Cell Active and Orally Bioavailable Tankyrase Inhibitors. |
|---|---|
| Release_Year | 2015 |
| PMID | 26396691 |
| DOI | 10.1021/acsmedchemlett.5b00251 |