PPIST10049
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | GSIQQATTGVSQETSENPGDKTIVPATLPQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQMIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMSLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPDMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQK |
Peptide Information
| Peptide_Chain | B |
|---|---|
| Peptide_Sequence | KENALLRYLLDKDD |
| Peptide_Length | 14 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 5G5W |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.20 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Discovery of Indazole Ethers as Novel, Potent, Non-Steroidal Glucocorticoid Receptor Modulators. |
|---|---|
| Release_Year | 2017 |
| PMID | 27810243 |
| DOI | 10.1016/J.BMCL.2016.10.052 |