PPIST11054

Protein Information
Protein_Chain A;C[auth B]
Protein_Sequence MHHHHHHSSGVDLGTENLYFQSMLNTSGSGTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAM
Peptide Information
Peptide_Chain B[auth I];D[auth J]
Peptide_Sequence KMAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPEG
Peptide_Length 49
Non-standard residues No
Interaction Information
PDB_ID 5NVH
Method X-RAY DIFFRACTION
Resolution 1.60 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title 2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors.
Release_Year 2018
PMID 29374194
DOI 10.1038/s41598-018-19872-3