PPIST11352

Protein Information
Protein_Chain A[auth B]/B[auth A]
Protein_Sequence QIQLVQSGPELKKPGETVKISCKASGYTFTDYSMHWVKQAPGKGLKWMGWINTATGEPTYADDFKGRFAFSLETSASTAYLQINNLKNEDTATYFCGRDYWGQGTTLTVSSAKTTPPSVYPLAPGCGDTTGSSVTLGCLVKGYFPESVTVTWNSGSLSSSVHTFPALLQSGLYTMSSSVTVPSSTWPSQTVTCSVAHPASSTTVDKKLEPS/DIQMIQSPSSLSASLGGKVTITCKASQDINKYIAWFQHKPGKGPTLLIYYTSTLQPGIPSRFSGSGSGRHYSFSISNLEPEDIATYYCLQYDNLRTFGGGTKLEIKRADAAPTVSIFPPSSEQLTSGGASVVCFLNNFYPKDINVKWKIDGSERQNGVLNSWTDQDSKDSTYSMSSTLTLTKDEYERHNSYTCEATHKTSTSPIVKSFNRNEC
Peptide Information
Peptide_Chain C
Peptide_Sequence SGRGKGGKGLGK
Peptide_Length 12
Non-standard residues No
Interaction Information
PDB_ID 5YE3
Method X-RAY DIFFRACTION
Resolution 1.70 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title JQ1 affects BRD2-dependent and independent transcription regulation without disrupting H4-hyperacetylated chromatin states.
Release_Year 2018
PMID 30080437
DOI 10.1080/15592294.2018.1469891