PPIST11722
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | MHNHNHNHNHNHNGGENLYFQGASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSGG |
Peptide Information
| Peptide_Chain | B[auth C] |
|---|---|
| Peptide_Sequence | KHKILHRLLQDS |
| Peptide_Length | 12 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 6ESN |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.84 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Potent and Orally Bioavailable Inverse Agonists of ROR gamma t Resulting from Structure-Based Design. |
|---|---|
| Release_Year | 2018 |
| PMID | 30095900 |
| DOI | 10.1021/acs.jmedchem.8b00783 |