PPIST12004
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | NTSGSGTILIDLSPDDKEFQSVEEEMQSTVREHRDGGHAGGIFNRYNILKIQKVCNKKLWERYTHRRKEVSEENHNHANERMLFHGSPFVNAIIHKGFDERHAYIGGMFGAGIYFAENSSKSNQYVYGIGGGTGCPVHKDRSCYICHRQLLFCRVTLGKSFLQFSAMK |
Peptide Information
| Peptide_Chain | B |
|---|---|
| Peptide_Sequence | MAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPEG |
| Peptide_Length | 48 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 5ZQO |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.06 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors. |
|---|---|
| Release_Year | 2019 |
| PMID | 30883102 |
| DOI | 10.1021/acs.jmedchem.8b01888 |