PPIST12886
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | IVGGTASVRGEWPWQVTLHTTSPTQRHLCGGSIIGNQWILTAAHCFYGVESPKILRVYSGILNQSEIKEDTSFFGVQEIIIHDQYKMAESGYDIALLKLETTVGYGDSQRPICLPSKGDRNVIYTDCWVTGWGYRKLRDKIQNTLQKAKIPLVTNEECQKRYRGHKITHKMICAGYREGGKDACKGDSGGPLSCKHNEVWHLVGITSWGEGCAQRERPGVYTNVVEYVDWILEKTQAVHHHHHH |
Peptide Information
| Peptide_Chain | B[auth H] |
|---|---|
| Peptide_Sequence | MDDDDKMDNECTTKIKPR |
| Peptide_Length | 18 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 5QTX |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.07 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Orally bioavailable amine-linked macrocyclic inhibitors of factor XIa. |
|---|---|
| Release_Year | 2020 |
| PMID | 31932224 |
| DOI | 10.1016/j.bmcl.2020.126949 |