PPIST14540
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | GSGFTSKDTYLSHFNPRDYLEKYYKFGSRHSAESQILKHLLKNLFKIFCLDGVKGDLLIDIGSGPTIYQLLSACESFKEIVVTDYSDQNLQELEKWLKKEPAAFDWSPVVTYVCDLEGNRVKGPEKEEKLRQAVKQVLKCDVTQSQPLGAVPLPPADCVLSTLCLDAACPDLPTYCRALRNLGSLLKPGGFLVIMDALKSSYYMIGEQKFSSLPLGREAVEAAVKEAGYTIEWFEVISQSYSSTMANNEGLFSLVARKL |
Peptide Information
| Peptide_Chain | B |
|---|---|
| Peptide_Sequence | GFPYKPXFC |
| Peptide_Length | 9 |
| Non-standard residues | Yes |
Interaction Information
| PDB_ID | 7EI2 |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.08 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Macrocyclic Peptides as a Novel Class of NNMT Inhibitors: A SAR Study Aimed at Inhibitory Activity in the Cell. |
|---|---|
| Release_Year | 2021 |
| PMID | 34267879 |
| DOI | 10.1021/acsmedchemlett.1c00134 |