PPIST14997
Protein Information
| Protein_Chain | A;B |
|---|---|
| Protein_Sequence | AMTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEKMSKDGKKKKKKSKTKCVIM |
Peptide Information
| Peptide_Chain | C[auth E];D[auth F] |
|---|---|
| Peptide_Sequence | AXPLYISYDPVCRA |
| Peptide_Length | 14 |
| Non-standard residues | Yes |
Interaction Information
| PDB_ID | 7ROV |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.32 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Discovery of cell active macrocyclic peptides with on-target inhibition of KRAS signaling. |
|---|---|
| Release_Year | 2021 |
| PMID | 35024121 |
| DOI | 10.1039/d1sc05187c |