PPIST15787

Protein Information
Protein_Chain A
Protein_Sequence EELQKSIGHKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGQAPIVNAPEGGKVDLEAFSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLACVERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPTELFPPLFLEVFED
Peptide Information
Peptide_Chain B
Peptide_Sequence ENALLRYLLDK
Peptide_Length 11
Non-standard residues No
Interaction Information
PDB_ID 7WML
Method X-RAY DIFFRACTION
Resolution 2.67 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title Discovery of a Highly Selective and H435R-Sensitive Thyroid Hormone Receptor beta Agonist.
Release_Year 2022
PMID 35507418
DOI 10.1021/acs.jmedchem.2c00144