PPIST16386
Protein Information
| Protein_Chain | A; D; G; J/C; F; I; L |
|---|---|
| Protein_Sequence | MDVFLMIRRHKTTIFTDAKESSTVFELKRIVEGILKRPPDEQRLYKDDQLLDDGKTLGECGFTSQTARPQAPATVGLAFRADDTFEALCIEPFSSPPELPDVMK/GSMEAGRPRPVLRSVNSREPSQVIFCNRSPRVVLPVWLNFDGEPQPYPTLPPGTGRRIHSYRGHLWLFRDAGTHDGLLVNQTELFVPSLNVDGQPIFANITLPVYTLKERCLQVVRSLVKPENYRRLDIVRSLYEDLEDHPNVQKDLERLTQERIAHQRMGD |
Peptide Information
| Peptide_Chain | B; E; H; K |
|---|---|
| Peptide_Sequence | MMYVKLISSDGHEFIVKREHALTSGTIKAMLSGPGQFAENETNEVNFREIPSHVLSKVCMYFTYKVRYTNSSTEIPEFPIAPEIALELLMAANFLDC |
| Peptide_Length | 97 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 8BDM |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.02 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Systematic Potency and Property Assessment of VHL Ligands and Implications on PROTAC Design. |
|---|---|
| Release_Year | 2023 |
| PMID | 36749883 |
| DOI | 10.1002/cmdc.202200615 |