PPIST16462
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | GPRSVASSKLWMLEFSAFLEQQQDPDTYNKHLFVHIGQSSPSYSDPYLEAVDIRQIYDKFPEKKGGLKDLFERGPSNAFFLVKFWADLNTNIEDEGSSFYGVSSQYESPENMIITCSTKVCSFGKQVVEKVETEYARYENGHYSYRIHRSPLCEYMINFIHKLKHLPEKYMMNSVLENFTILQVVTNRDTQETLLCIAYVFEVSASEHGAQHHIYRLVKE |
Peptide Information
| Peptide_Chain | B |
|---|---|
| Peptide_Sequence | XFSPADFHXDIACDVARGX |
| Peptide_Length | 19 |
| Non-standard residues | Yes |
Interaction Information
| PDB_ID | 8C17 |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 2.25 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Biochemical and Structural Characterization of a Peptidic Inhibitor of the YAP:TEAD Interaction That Binds to the alpha-Helix Pocket on TEAD. |
|---|---|
| Release_Year | 2023 |
| PMID | 36825662 |
| DOI | 10.1021/acschembio.2c00936 |