PPIST16978

Protein Information
Protein_Chain A
Protein_Sequence VDESKKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPSNCQNKESASKQS
Peptide Information
Peptide_Chain B
Peptide_Sequence GSVSSVPTKLEVVAATPTSLLISWDAQTYQMYDYVSYYRITYGETGGNSPVQEFTVPGYYSTATISGLKPGVDYTITVYAEGYYSSYSPISINYRT
Peptide_Length 96
Non-standard residues No
Interaction Information
PDB_ID 8SSP
Method X-RAY DIFFRACTION
Resolution 2.60 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title A biophysical framework for double-drugging kinases.
Release_Year 2023
PMID 37590418
DOI 10.1073/pnas.2304611120