PPIST17333
Protein Information
| Protein_Chain | A |
|---|---|
| Protein_Sequence | SMTSSANEDMPVERILEAELAVEPKTETYVEANMGLNPSSPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQMT |
Peptide Information
| Peptide_Chain | B |
|---|---|
| Peptide_Sequence | KHKILHRLLQDSSY |
| Peptide_Length | 14 |
| Non-standard residues | No |
Interaction Information
| PDB_ID | 8PP0 |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.90 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Structure-Guided Design of a Highly Potent Partial RXR Agonist with Superior Physicochemical Properties. |
|---|---|
| Release_Year | 2024 |
| PMID | 38237049 |
| DOI | 10.1021/acs.jmedchem.3c02095 |