PPIST17503

Protein Information
Protein_Chain A;B;C
Protein_Sequence MGSSHHHHHHSSGLVPRGSHMDPNSLRHKYNFIADVVEKIAPAVVHIELFRKLPFSKREVPVASGSGFIVSEDGLIVTNAHVVTNKHRVKVELKNGATYEAKIKDVDEKADIALIKIDHQGKLPVLLLGRSSELRPGEFVVAIGSPFSLQNTVTTGIVSTTQRGGKELGLRNSDMDYIQTDAIINYGNAGGPLVNLDGEVIGINTLKVTAGISFAIPSDKIKKFLTESHDRQAKGKAITK
Peptide Information
Peptide_Chain D[auth I];E[auth X];F[auth Y]
Peptide_Sequence HADPICNKPCKTHDDCSGAWFCQACYYATWSCGPYVG
Peptide_Length 37
Non-standard residues No
Interaction Information
PDB_ID 8SDM
Method X-RAY DIFFRACTION
Resolution 3.05 angstrom
Structure
Protein-peptide residue interaction
Residues
Acidic
Polar
Basic
Aliphatic
Aromatic
Interactions
HBond
WaterBridge
Hydrophobic
SaltBridge
PiStack
PiCation
Halogen
Metal
Interaction_xlsx Download interaction table (.xlsx)
Reference Information
Title Cystine-knot peptide inhibitors of HTRA1 bind to a cryptic pocket within the active site region.
Release_Year 2024
PMID 38777835
DOI 10.1038/s41467-024-48655-w