PPIST17733
Protein Information
| Protein_Chain | A;B |
|---|---|
| Protein_Sequence | AAHLSDMLQQLHSVNASKPSERGLVRQEEAEDPACIPIFWVSKWVDYSDKYGLGYQLCDNSVGVLFNDSTRLILYNDGDSLQYIERDGTESYLTVSSHPNSLMKKITLLKYFRNYMSEHLLKAGANITPREGDELARLPYLRTWFRTRSAIILHLSNGSVQINFFQDHTKLILCPLMAAVTYIDEKRDFRTYRLSLLEEYGCCKELASRLRYARTMVDKLLSSRSA |
Peptide Information
| Peptide_Chain | C;D |
|---|---|
| Peptide_Sequence | XPLHSTX |
| Peptide_Length | 7 |
| Non-standard residues | Yes |
Interaction Information
| PDB_ID | 8WFP |
|---|---|
| Method | X-RAY DIFFRACTION |
| Resolution | 1.99 angstrom |
| Structure | |
| Protein-peptide residue interaction | |
| Interaction_xlsx | Download interaction table (.xlsx) |
Reference Information
| Title | Degradation of Polo-like Kinase 1 by the Novel Poly-Arginine N-Degron Pathway PROTAC Regulates Tumor Growth in Nonsmall Cell Lung Cancer. |
|---|---|
| Release_Year | 2024 |
| PMID | 38105611 |
| DOI | 10.1021/acs.jmedchem.3c01493 |