|
PPIRE01545 |
IC50=3.8 nM |
RGDYK |
|
PPIRE02045 |
IC50=0.21 uM |
EGKRGDfKRGDf |
|
PPIRE02046 |
IC50=0.32 uM |
EGKRGDfKRGDf |
|
PPIRE02047 |
IC50=0.63 uM |
EGKRGDfKRGDf |
|
PPIRE03671 |
IC50=10000 nM |
RGDfX |
|
PPIRE03672 |
IC50=2000 nM |
RGDfX |
|
PPIRE03673 |
IC50=10000 nM |
RGDfX |
|
PPIRE03674 |
IC50=10000 nM |
RGDfX |
|
PPIRE03675 |
IC50=500 nM |
RGDX |
|
PPIRE03676 |
IC50=8 nM |
RGDX |
|
PPIRE04736 |
KD=9.03 uM |
AGDV |
|
PPIRE04737 |
KD=1 uM |
AGDV |
|
PPIRE04738 |
KD=50.6 uM |
AGDV |
|
PPIRE04739 |
KD=67.7 uM |
AGDV |
|
PPIRE04740 |
KD=216.7 uM |
AGDv |
|
PPIRE05069 |
Ki=62 uM |
RGDS |
|
PPIRE05362 |
IC50=1.49 mM |
RGDX |
|
PPIRE05516 |
IC50=0.56 mM |
GRGDS |
|
PPIRE05722 |
KD=7.85 uM |
QAGDV |
|
PPIRE06061 |
IC50=422 nM |
RGDfK |
|
PPIRE06070 |
IC50=1.33 nM |
RGDfK |
|
PPIRE06071 |
IC50=0.94 nM |
RGDfK |
|
PPIRE06072 |
IC50=1.02 nM |
RGDfK |
|
PPIRE06073 |
IC50=0.51 nM |
RGDfK |
|
PPIRE06080 |
IC50=47.1 nM |
RGDfX |
|
PPIRE06083 |
IC50=98.1 uM |
RGDVX |
|
PPIRE06089 |
IC50=597 uM |
RGDXX |
|
PPIRE06091 |
IC50=3.2 nM |
RGDXX |
|
PPIRE06093 |
IC50=1816 nM |
RGDXX |
|
PPIRE06095 |
IC50=53.7 nM |
RGDXX |
|
PPIRE06097 |
IC50=88 nM |
RGDXX |
|
PPIRE06099 |
IC50=460 nM |
RGDXX |
|
PPIRE06101 |
IC50=10000 nM |
RGDXX |
|
PPIRE06103 |
IC50=114 nM |
RGDXX |
|
PPIRE06105 |
IC50=10000 nM |
RGDXX |
|
PPIRE06107 |
IC50=1850 nM |
RGDXX |
|
PPIRE06110 |
IC50=42.2 nM |
RGDYK |
|
PPIRE06111 |
IC50=40.02 nM |
RGDYK |
|
PPIRE06315 |
KD=0.41 uM |
GRGDSP |
|
PPIRE06317 |
KD=1.6 uM |
GRGDSP |
|
PPIRE06566 |
IC50=12 uM |
RGDFDV |
|
PPIRE06570 |
IC50=2200 uM |
RGYFDV |
|
PPIRE06774 |
IC50=414 nM |
cRGDfK |
|
PPIRE06815 |
IC50=0.67 uM |
RGDDYK |
|
PPIRE06930 |
IC50=1.7 nM |
RGDfX |
|
PPIRE06978 |
IC50=9.71 nM |
RGDfX |
|
PPIRE06990 |
IC50=30.4 nM |
RGDfX |
|
PPIRE06991 |
IC50=2.99 nM |
RGDfX |
|
PPIRE07023 |
IC50=9.38 nM |
RGDfX |
|
PPIRE07027 |
IC50=3 nM |
RGDfX |
|
PPIRE07080 |
IC50=1.08 nM |
RGDtX |
|
PPIRE07081 |
IC50=11 nM |
RGDtX |
|
PPIRE07094 |
IC50=4.36 nM |
RGDtX |
|
PPIRE07145 |
IC50=6.2 nM |
RGDtX |
|
PPIRE07189 |
Ka=7.00E+06 1/M |
CDCRGDCFC |
|
PPIRE07191 |
IC50=7 nM |
CDCRGDCFC |
|
PPIRE07197 |
IC50=309 nM |
CVRGDF |
|
PPIRE07200 |
IC50=29 nM |
CVRGDF |
|
PPIRE07392 |
IC50=20 nM |
CVRGDFC |
|
PPIRE07898 |
KD=2.412 nM |
RGDFRWPR |
|
PPIRE08452 |
IC50=100 uM |
GIDLTSLTK |
|
PPIRE08474 |
KD=2.3 uM |
GRGDLGRLK |
|
PPIRE08662 |
IC50=1.8 nM |
RGDfK |
|
PPIRE08706 |
IC50=0.5 uM |
RGDLADLRK |
|
PPIRE08711 |
IC50=2.2 uM |
RGDLMKLAK |
|
PPIRE08716 |
IC50=0.3 uM |
RGDLRELAK |
|
PPIRE08782 |
KD=2.5 uM |
RRGDLATIH |
|
PPIRE08848 |
KD=4.8 uM |
TSGDQKTIK |
|
PPIRE08853 |
IC50=3.2 nM |
RGDtV |
|
PPIRE08860 |
IC50=100 uM |
VGDLTYLKK |
|
PPIRE08897 |
IC50=100000 nM |
DGRKfDGRKfDGRKf |
|
PPIRE08977 |
IC50=43 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09006 |
IC50=44 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09007 |
IC50=50 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09008 |
IC50=74 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09009 |
IC50=85 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09010 |
IC50=56 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09011 |
IC50=125 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09012 |
IC50=240 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09013 |
IC50=220 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09014 |
IC50=56 nM |
RGDfKRGDfKRGDfK |
|
PPIRE09015 |
Ki=1.63 nM |
RGDfKERGDfK |
|
PPIRE09016 |
Ki=1.56 nM |
RGDfKERGDfK |
|
PPIRE09017 |
Ki=3.01 nM |
RGDfKERGDfK |
|
PPIRE09018 |
Ki=1.21 nM |
RGDfKERGDfK |
|
PPIRE09087 |
IC50=25 nM |
ERGDfKRGDfK |
|
PPIRE09210 |
IC50=9.9 nM |
RGDfX |
|
PPIRE09211 |
IC50=5.5 nM |
RGDfX |
|
PPIRE09308 |
IC50=72 nM |
RGDfX |
|
PPIRE09391 |
IC50=11 nM |
RGDfX |
|
PPIRE09392 |
IC50=3.3 nM |
RGDfX |
|
PPIRE09591 |
IC50=700 uM |
RQMIRGYFDV |
|
PPIRE10271 |
KD=15.28 nM |
ERGDFKRGDFK |
|
PPIRE10274 |
IC50=102 nM |
ERGDfKRGDfK |
|
PPIRE10295 |
IC50=85 nM |
RGDfKERGDfK |
|
PPIRE10297 |
KD=15.07 nM |
ERGDfKRGDfK |
|
PPIRE10562 |
KD=0.64 uM |
HHLGGAKQAGDV |
|
PPIRE10563 |
KD=1.27 uM |
HHLGGAKQAGDV |
|
PPIRE10877 |
IC50=23.9 nM |
ECRGDfK |
|
PPIRE10878 |
IC50=26.6 nM |
ECRGDfK |
|
PPIRE11032 |
IC50=8.99 nM |
ECRGDfKCRGDfK |
|
PPIRE11035 |
IC50=3.34 nM |
ECRGDfKCRGDfK |
|
PPIRE11054 |
IC50=1.74 nM |
EECRGDfKCRGDfKECRGDfKCRGDfK |
|
PPIRE11107 |
IC50=1.8 nM |
EECRGDfKCRGDfKECRGDfKCRGDfK |
|
PPIRE11147 |
IC50=120 nM |
ERGDfK |
|
PPIRE11148 |
IC50=69.9 nM |
ERGDfKRGDfK |
|
PPIRE11149 |
IC50=19.6 nM |
EERGDfKRGDfKERGDfKRGDfK |
|
PPIRE11307 |
IC50=29 nM |
EcRGDfXcRGDfX |
|
PPIRE11308 |
IC50=27 nM |
EcRGDfXcRGDfX |
|
PPIRE11330 |
IC50=21.67 nM |
RGDYKEATWLPPR |
|
PPIRE11337 |
IC50=32 nM |
XRGDfKXRGDfKX |
|
PPIRE11338 |
IC50=39 nM |
XRGDfKXRGDfKX |
|
PPIRE11670 |
IC50=74 nM |
XEXRGDfKXRGDfK |
|
PPIRE12137 |
IC50=596 nM |
EcRGKXfdcRGKXfd |
|
PPIRE13251 |
IC50=10 uM |
NAVPNLRGDLQVLAQRVART |
|
PPIRE13348 |
IC50=1.1 nM |
GGGEGGGRGDfKGGGRGDfK |
|
PPIRE13349 |
IC50=62 nM |
GGGEGGGRGDfKGGGRGDfK |
|
PPIRE13667 |
IC50=10 nM |
EERGDfKRGDfKERGDfKRGDfK |
|
PPIRE13674 |
KD=50 uM |
KVGFFKRNRNSPPVNELLEEDQGQ |
|
PPIRE13675 |
KD=7.7 uM |
KVGFFKRNRNSPPVNELLEEDQGQ |
|
PPIRE13718 |
IC50=1.4 nM |
EERGDfKRGDfKEERGDfKRGDfK |
|
PPIRE13884 |
KD=131.6 nM |
TMPFLFCNVNDVCNFASRNDYSKKK |
|
PPIRE13963 |
IC50=71.7 nM |
RGDfK |
|
PPIRE13978 |
IC50=35.2 nM |
RGDfK |
|
PPIRE14725 |
IC50=0.4 nM |
EGGGEGGGRGDfKGGGRGDfKEGGGEGGGRGDfKGGGRGDfK |
|
PPIRE14840 |
KD=160 nM |
XXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXXX |
|
PPIRE14998 |
IC50=1 nM |
RGDfK |
|
PPIRE14999 |
IC50=0.1 nM |
ERGDfKRGDfK |
|
PPIRE15009 |
IC50=3.6 nM |
EFECESGPCCRNCKFLKEGTICKRARGDDMDDYCNGKTCDCPRNPHKGPAT |
|
PPIRE15010 |
IC50=5 mM |
PRNPHKGPAT |
|
PPIRE15011 |
IC50=5 mM |
APRNPHKGPAT |
|
PPIRE15022 |
IC50=0.5 nM |
RGDfKRGDfK |
|
PPIRE15040 |
KD=30 uM |
RGDfV |
|
PPIRE15041 |
KD=5.05 uM |
RGDfV |
|
PPIRE15042 |
Ki=42 uM |
RGDfV |
|
PPIRE15043 |
IC50=29 uM |
RGDfV |
|
PPIRE15044 |
IC50=230 nM |
RGDfV |
|
PPIRE15045 |
IC50=12 uM |
RGDfV |
|
PPIRE15046 |
KD=1 mM |
RGD |
|
PPIRE15047 |
Ki=21 uM |
RGDS |
|
PPIRE15048 |
Ki=293 uM |
RGDS |
|
PPIRE15057 |
IC50=0.37 uM |
RGDfXV |
|
PPIRE15058 |
IC50=2.69 uM |
RGDfXV |
|
PPIRE15060 |
IC50=0.076 uM |
RGDfXV |
|
PPIRE15061 |
IC50=0.44 uM |
RGDfXV |
|
PPIRE15062 |
IC50=0.42 uM |
RGDfXV |
|
PPIRE15063 |
IC50=3.62 uM |
RGDfXV |
|
PPIRE15065 |
IC50=0.036 uM |
RGDfXV |
|
PPIRE15066 |
IC50=0.14 uM |
RGDfXV |
|
PPIRE15067 |
IC50=12.42 uM |
RGDfXV |
|
PPIRE15068 |
IC50=171.5 uM |
RGDfXV |
|
PPIRE15069 |
IC50=1.38 uM |
RGDfXV |
|
PPIRE15070 |
IC50=4.55 uM |
RGDfXV |
|
PPIRE15071 |
IC50=22.3 uM |
RGDfXV |
|
PPIRE15072 |
IC50=143.1 uM |
RGDfXV |
|
PPIRE15073 |
IC50=0.28 uM |
RGDfXV |
|
PPIRE15074 |
IC50=2.31 uM |
RGDfXV |
|
PPIRE15078 |
IC50=440 nM |
RGDyX |
|
PPIRE15082 |
IC50=432 nM |
RGDyX |
|
PPIRE15083 |
IC50=3.4 nM |
RGDyX |
|
PPIRE15084 |
IC50=7.1 nM |
RGDyX |
|
PPIRE15085 |
IC50=242 nM |
RGDyX |
|
PPIRE15086 |
IC50=866 nM |
RGDyX |
|
PPIRE15251 |
KD=185 nM |
FRGDLMQL |
|
PPIRE16549 |
IC50=43 uM |
RGDF |
|
PPIRE16550 |
IC50=20 uM |
RGDW |
|
PPIRE16551 |
IC50=200 uM |
RGDS |
|
PPIRE16689 |
IC50=1000 nM |
XXGRG |
|
PPIRE16692 |
IC50=10000 nM |
XXGRG |
|
PPIRE16694 |
IC50=516 nM |
XXGRK |
|
PPIRE16697 |
IC50=10000 nM |
XXGRK |
|
PPIRE16699 |
IC50=10000 nM |
XXGRk |
|
PPIRE16702 |
IC50=10000 nM |
XXGRk |
|
PPIRE16704 |
IC50=10000 nM |
XXGRw |
|
PPIRE16707 |
IC50=10000 nM |
XXGRw |
|
PPIRE16717 |
IC50=0.68 pM |
CRGDC |
|
PPIRE16718 |
IC50=100 pM |
CRGdC |
|
PPIRE18920 |
IC50=5 uM |
GRGDS |
|
PPIRE18921 |
IC50=0.16 uM |
RGDfK |
|
PPIRE18922 |
IC50=100 uM |
FYFDLRK |
|
PPIRE18975 |
IC50=0.46 uM |
cGRGDdvc |
|
PPIRE18976 |
IC50=20 uM |
CGRGDdvC |
|
PPIRE18977 |
IC50=1.84 uM |
cGRGDdic |
|
PPIRE18978 |
IC50=0.07 uM |
cGRGDdXc |
|
PPIRE18979 |
IC50=0.13 uM |
cGRGDdXc |
|
PPIRE18980 |
IC50=0.09 uM |
cGRGDdXc |
|
PPIPT00580 |
IC50=6.22 nM |
RGDYKE |
|
PPIPT00583 |
IC50=1.69 uM |
RGDYKE |
|
PPIPT00584 |
IC50=18 nM |
RGDFKE |
|
PPIPT00587 |
IC50=6.01 uM |
RGDFKE |
|
PPIPT00770 |
IC50=860 nM |
CRGDfK |
|
PPIPT00771 |
IC50=370 nM |
GCWTGRGDSPASSCKQDSDCLAGCWCGPNGFCG |
|
PPIPT00772 |
IC50=16 nM |
GCHPPRGDNPPWTCKQDSDCLAGCVCGPNGFCG |
|
PPIPT00773 |
IC50=26 nM |
GCPQGRGDWAPTSCKQDSDCRAGCVCGPNGFCG |
|
PPIPT00774 |
IC50=2.6 nM |
GCHWGRGDWAPEECKQDSDCOAGCWCGPNGFCG |
|
PPIPT00775 |
KD=0.89 nM |
GCVRLHESCLGOOVPCCDPAATCYCSGRGDNDLWCYCR |
|
PPIPT00776 |
KD=18 nM |
GCVRLHESCLGOOVPCCDPAATCYCWGRGDDNLKCYCR |
|
PPIPT00777 |
KD=24 nM |
GCVRLHESCLGOOVPCCDPAATCYCKGRGDARLQCYCR |
|
PPIPT00778 |
KD=1.6 nM |
GCVRLHESCLGOOVPCCDPAATCYCEGRGDRDMKCYCR |
|
PPIPT00929 |
KD=2.1 nM |
GCVRLHESCLGQQVPCCDPAATCYCSGRGDNDLWCYCR |
|
PPIPT00930 |
KD=4.6 nM |
GCHPPRGDNPPVTCKOSDSDCLAGCVCGPNGFCGSP |
|
PPIPT00931 |
KD=1.72 nM |
GCPOGRGDWAPTSCKOSDSDCLAGCVCGPNGFCGSP |
|
PPIPT01094 |
IC50=3.4 nM |
HHLLHK |
|
PPIPT01095 |
IC50=30.7 nM |
HGDLHK |
|
PPIPT01096 |
IC50=2.43 nM |
HHDLHK |
|
PPIPT01097 |
IC50=46 nM |
HGLVHK |
|
PPIPT01098 |
IC50=313 nM |
HSLVHK |
|
PPIPT01099 |
IC50=44.7 nM |
HHLVHK |
|
PPIPT01100 |
IC50=1.74 nM |
HGDVHK |
|
PPIPT01221 |
KD=1.72 nM |
GCPQGRGDWAPTSCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01386 |
IC50=370 nM |
GCVTGRGDSPASSCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01387 |
IC50=62.9 nM |
GCAEPRGDMPWTWCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01388 |
IC50=33.9 nM |
GCVQGRGDWSPPSCKQDSDCPAGCVCGPNGFCG |
|
PPIPT01389 |
IC50=13 nM |
GCPRPRGDNPPLTCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01416 |
IC50=860 nM |
CRGDYK |
|
PPIPT01417 |
IC50=370 nM |
GCTGRGDSPASSKCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01418 |
IC50=13 nM |
GCTIGRGDWAPSECKQDSDCLAGCVCGPNGFCG |
|
PPIPT01419 |
IC50=16 nM |
GCPQGRGDWAPTSCKQDSDCRAGCVCGPNGFCG |
|
PPIPT01420 |
IC50=26 nM |
GCPRPRGDNPPLTCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01512 |
IC50=6.1 nM |
GCTIGRGDWAPSECKQDSDCLAGCWCGPNGFCG |
|
PPIPT01513 |
IC50=26 nM |
GCPQGRGDWAPTSCKQDSDCRAGCVCGPNGFCG |
|
PPIPT01514 |
IC50=62.9 nM |
GCPRPRGDNPPLTCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01515 |
IC50=1333 nM |
GCTGRGDSSPASSKCKQDSDCLAGCVCGPNGFCG |
|
PPIPT01516 |
IC50=860 nM |
CDCRGDfK |
|
PPIPT01721 |
KD=0.78 nM |
GCVRLHESCLGQQVPCCDPAATCYCSGRGDNDLVCYCR |
|
PPIPT01722 |
KD=0.89 nM |
GCVRLHESCLGQQVPCCDPAATCYCSGRGDNDLVCYCR |
|
PPIPT02014 |
IC50=8.4 nM |
aRGDAA |
|
PPIPT02015 |
IC50=0.6 nM |
VRGDAA |
|
PPIPT02366 |
IC50=1000 uM |
CSGRCGVRY |
|
PPIPT02367 |
IC50=1000 uM |
CNGRCGVRY |
|
PPIPT02368 |
IC50=25 uM |
CDGRCGVRY |
|
PPIPT02369 |
IC50=0.5 uM |
CXGRCGVRY |
|
PPIPT02370 |
IC50=0.1 uM |
cXGRCGVRY |
|
PPIPT02381 |
KD=100 nM |
CDCRGDCFC |