PPIDT00424

Drug Information
NameTirzepatide
SequenceYXEGTFTSDYSIXLDKIAQKAFVQWLIAGGPSSGAPPPS
DrugBank_IDDB15171
Typebiotech
IndicationTirzepatide is indicated as an adjunct to diet and exercise to improve glycemic control in adults with type 2 diabetes mellitus or for the chronic weight management for adult patients that are obese or overweight with at least one weight-related comorbid condition such as hypertension, dyslipidemia, type 2 diabetes mellitus, obstructive sleep apnea, or cardiovascular disease). [L41815,L44376,L48761] In Europe, it may be used as monotherapy or in combination with other drugs used to treat diabetes.[L44376] This drug has not been studied in patients with a history of pancreatitis. Tirzepatide is not indicated for use in patients with type 1 diabetes mellitus.[L41815]

Dosage Forms
Form Route Strength
Injection, solution Subcutaneous
10 mg/0.5mL
Injection, solution Subcutaneous
10 mg
Injection, solution Subcutaneous
10 mg/dose
Injection, solution Subcutaneous
12.5 mg/dose
Injection, solution Subcutaneous
12.5 mg/0.5mL
Injection, solution Subcutaneous
12.5 mg
Injection, solution Subcutaneous
15 mg
Injection, solution Subcutaneous
15 mg/0.5mL
Injection, solution Subcutaneous
15 mg/dose
Injection, solution Subcutaneous
2.5 mg/dose
Injection, solution Subcutaneous
2.5 mg
Injection, solution Subcutaneous
2.5 mg/0.5mL
Injection, solution Subcutaneous
5 mg/dose
Injection, solution Subcutaneous
5 mg/0.5mL
Injection, solution Subcutaneous
5 mg
Injection, solution Subcutaneous
7.5 mg/0.5mL
Injection, solution Subcutaneous
7.5 mg
Injection, solution Subcutaneous
7.5 mg/dose
Solution Subcutaneous
10 mg / 0.5 mL
Solution Subcutaneous
12.5 mg / 0.5 mL
Solution Subcutaneous
15 mg / 0.5 mL
Solution Subcutaneous
2.5 mg / 0.5 mL
Solution Subcutaneous
5 mg / 0.5 mL
Solution Subcutaneous
7.5 mg / 0.5 mL
Solution Subcutaneous
10 mg
Solution Subcutaneous
12.5 mg
Solution Subcutaneous
15 mg
Solution Subcutaneous
2.5 mg
Solution Subcutaneous
5 mg
Solution Subcutaneous
7.5 mg
Solution Subcutaneous
10 mg / 0.6 mL
Solution Subcutaneous
12.5 mg / 0.6 mL
Solution Subcutaneous
15 mg / 0.6 mL
Solution Subcutaneous
2.5 mg / 0.6 mL
Solution Subcutaneous
5 mg / 0.6 mL
Solution Subcutaneous
7.5 mg / 0.6 mL
10 mg/dose
15 mg/dose
Target Information
Role Uniprot_ID Gene_Name Entity_Name Organism Actions Internal link
target P43220 GLP1R Glucagon-like peptide 1 receptor Homo sapiens agonist Link
target P48546 GIPR Gastric inhibitory polypeptide receptor Homo sapiens agonist Link
carrier P02768 ALB Albumin Homo sapiens binder Link