|
PPIRE01907 |
IC50=669 nM |
HXEGTXTSDXX |
|
PPIRE02894 |
IC50=0.4 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE02895 |
IC50=22 nM |
HXEGXFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE02896 |
IC50=7.8 nM |
HxEGXFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE02897 |
IC50=0.6 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE02898 |
IC50=6.5 nM |
HXEGXFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE02899 |
IC50=11 nM |
HXEGXFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE02900 |
IC50=3 nM |
HXEGXFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE02901 |
IC50=1.5 nM |
HxEGXFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE14223 |
IC50=43.4 nM |
HAEGTFTNDMTNYLEEKAAKEFVGWLINGR |
|
PPIRE14224 |
IC50=1.1 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE14230 |
IC50=1 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE14232 |
IC50=1.1 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE14234 |
IC50=0.37 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE14249 |
IC50=1.1 nM |
HAEGTYTNDVTEYLEEKAAKEFIEWLIKGK |
|
PPIRE14253 |
IC50=81.1 nM |
HVEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE14254 |
IC50=4.76 nM |
HXEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE14272 |
IC50=10.9 nM |
DLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE14273 |
IC50=48.1 nM |
DLSKQMEEEAVRLFIEWLXNGGPSSGAPPPS |
|
PPIRE14274 |
IC50=137.2 nM |
DLSKQMEEEAVRLFIEWLXNGGPSSGAPPPS |
|
PPIRE14275 |
IC50=143.3 nM |
DLSKQMEEEAVRLFIEWLXNGGPSSGAPPPS |
|
PPIRE14316 |
IC50=44.1 nM |
DLSKQMEEEAVRLFIEWLKNGGPSSGAPPPSX |
|
PPIRE14317 |
IC50=29.7 nM |
DLSKQMEEEAVRLFIEWLKNGGPSSGAPPPSX |
|
PPIRE14318 |
IC50=46.7 nM |
DLSKQMEEEAVRLFIEWLKNGGPSSGAPPPSX |
|
PPIRE14326 |
IC50=17.5 nM |
HAEGTFTSDVTQQLDEKAAKEFIDWLINGGPS |
|
PPIRE14327 |
IC50=2.9 nM |
HAEGTYTNDVTEYLEEKAAKEFIEWLIKGKPK |
|
PPIRE14586 |
IC50=12.7 nM |
HAEGTFTSDVTQQLDEKAAKEFIDWLINGGPSKEIIS |
|
PPIRE14633 |
IC50=0.3708 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE14634 |
IC50=0.76 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE14684 |
IC50=0.9 nM |
HGEGTFTSDLSKQXEEEAVRLFIEWLKNGGPSSGAPPPSX |
|
PPIRE16787 |
EC50=1.2 nM |
HSEGTFTSDVSSYLEGQAAKEFIAWLVKGGVKALIDEILAA |
|
PPIRE16788 |
EC50=0.13 nM |
HSEGTFTSDVSSYLEGQAAKEFIAWLVKGGVKALIDEILAA |
|
PPIRE16789 |
IC50=12 nM |
HSEGTFTSDVSSYLEGQAAKEFIAWLVKGGVKALIDEILAA |
|
PPIRE17042 |
KD=116 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE17043 |
KD=99 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE17044 |
KD=180 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE17045 |
KD=1 uM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE17046 |
KD=1.1 uM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIRE17797 |
EC50=0.16 nM |
HGEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE17798 |
EC50=0.06 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIRE18566 |
EC50=1.8 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIRE18719 |
IC50=0.36 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIRE18720 |
IC50=4.5 nM |
LSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIPT00576 |
EC50=10 nM |
HEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT00577 |
EC50=0.204 nM |
QHAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT00578 |
EC50=0.312 nM |
AHAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT00835 |
EC50=5 nM |
RGKVLWAIFEKAAQGELYSSVDSTFTGEAH |
|
PPIPT00836 |
EC50=30 nM |
RGKVLWaIFEKAAQGELYSSVDSTFTGEAH |
|
PPIPT00837 |
EC50=1 nM |
RGKVLWEIFEKAAQGEKYSSEDSTFTGEaH |
|
PPIPT00838 |
EC50=1 nM |
RGKVLWEIFEKAAQKELYESVDSTFTGEaH |
|
PPIPT01279 |
EC50=10 nM |
HEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT01280 |
EC50=0.204 nM |
QHAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT01281 |
EC50=0.312 nM |
AHAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT01282 |
EC50=0.147 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT01283 |
EC50=120 nM |
AHAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT01284 |
EC50=135 nM |
QHAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT01285 |
EC50=2560 nM |
AEGTFTSDVSSYLEGQAAKEFIAWLVKGRG |
|
PPIPT02140 |
EC50=420 nM |
HXIGTMeFTSD |
|
PPIPT02142 |
EC50=59 nM |
HQGTTFTTSTDTYSKYLDTS |
|
PPIPT02143 |
EC50=12 uM |
HQGTTFTTSTDTYSKYLDTS |
|
PPIPT02144 |
EC50=11 uM |
HQGTTFTTSTDTYSKYLDTS |
|
PPIPT02145 |
EC50=0.009 nM |
HXIGTMeFTSD |
|
PPIPT02146 |
EC50=0.005 nM |
HXIGTMeFTSD |
|
PPIPT02148 |
EC50=0.007 nM |
HXIGTMeFTSD |
|
PPIPT02421 |
KD=420 nM |
HXQGTFTSDYSKYLDEQAAKEFIKWLLQT |
|
PPIPT02566 |
IC50=3.7 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02567 |
IC50=41 nM |
HAEGTFTGDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02568 |
IC50=22 nM |
HAEGTFTXSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02569 |
IC50=236 nM |
HAEGTFTSXXXXDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02570 |
IC50=400 nM |
HAEGTFTSXXXXXXXXDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02704 |
IC50=3.7 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02705 |
IC50=41 nM |
HGEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02706 |
IC50=22 nM |
HAXEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02707 |
IC50=44.9 nM |
HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR |
|
PPIPT02708 |
IC50=129 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIPT02709 |
IC50=34.5 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAP |
|
PPIPT02710 |
IC50=21.2 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGA |
|
PPIPT02711 |
IC50=3.22 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSS |
|
PPIPT02712 |
IC50=8.8 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGP |
|
PPIPT02713 |
IC50=7.0 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGG |
|
PPIPT02761 |
IC50=3.7 nM |
HAEGTFTSDWSSYLEGQAAKEFIAWLWKGRG |
|
PPIPT02762 |
IC50=41 nM |
GHAEGTFTSDWSSYLEGQAAKEFIAWLWKGRG |
|
PPIPT02763 |
IC50=34.5 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAPPPS |
|
PPIPT02764 |
IC50=21.2 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGAP |
|
PPIPT02765 |
IC50=3.2 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGA |
|
PPIPT02766 |
IC50=8.8 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPS |
|
PPIPT02767 |
IC50=7.0 nM |
HGEGTFTSDLSKQMEEEAVRLFIEWLKNGG |